SLC22A1 (solute carrier family 22 member 1)

2010-05-01  

Identity

HGNC
LOCATION
6q25.3
LOCUSID
ALIAS
HOCT1,OCT1,oct1_cds
FUSION GENES

Other Information

Locus ID:

NCBI: 6580
MIM: 602607
HGNC: 10963
Ensembl: ENSG00000175003

Variants:

dbSNP: 6580
ClinVar: 6580
TCGA: ENSG00000175003
COSMIC: SLC22A1

RNA/Proteins

Gene IDTranscript IDUniprot
ENSG00000175003ENST00000324965O15245
ENSG00000175003ENST00000366963O15245
ENSG00000175003ENST00000457470O15245
ENSG00000175003ENST00000460902O15245
ENSG00000175003ENST00000539263F5H5P3
ENSG00000175003ENST00000540443F5GY86

Expression (GTEx)

0
50
100
150
200
250
300
350
400

Pathways

PathwaySourceExternal ID
Bile secretionKEGGko04976
Bile secretionKEGGhsa04976
Choline metabolism in cancerKEGGhsa05231
Choline metabolism in cancerKEGGko05231
Neuronal SystemREACTOMER-HSA-112316
Transmission across Chemical SynapsesREACTOMER-HSA-112315
Neurotransmitter Release CycleREACTOMER-HSA-112310
Norepinephrine Neurotransmitter Release CycleREACTOMER-HSA-181430
Neurotransmitter Clearance In The Synaptic CleftREACTOMER-HSA-112311
Transmembrane transport of small moleculesREACTOMER-HSA-382551
SLC-mediated transmembrane transportREACTOMER-HSA-425407
Transport of glucose and other sugars, bile salts and organic acids, metal ions and amine compoundsREACTOMER-HSA-425366
Na+/Cl- dependent neurotransmitter transportersREACTOMER-HSA-442660
Organic cation/anion/zwitterion transportREACTOMER-HSA-549132
Organic cation transportREACTOMER-HSA-549127
MetabolismREACTOMER-HSA-1430728
Abacavir transport and metabolismREACTOMER-HSA-2161522
Abacavir transmembrane transportREACTOMER-HSA-2161517

Protein levels (Protein atlas)

Not detected
Low
Medium
High

PharmGKB

Entity IDNameTypeEvidenceAssociationPKPDPMIDs
PA10804imatinibChemicalClinicalAnnotation, VipGeneassociatedPKPD19584153, 23223357, 18398725, 24589908, 28762371, 29427770, 30237583, 30713339
PA151958383Gastrointestinal Stromal TumorsDiseaseClinicalAnnotationassociatedPD28762371
PA161925594tropisetronChemicalVipGeneassociated20921968
PA164712420AnticholinergicsChemicalClinicalAnnotationassociatedPD
PA164712431Antiemetics And AntinauseantsChemicalVariantAnnotationassociatedPKPD20921968
PA164712697Dopamine agonistsChemicalClinicalAnnotationassociatedPD
PA166129521sedationDiseaseVariantAnnotationassociatedPD23835420
PA166131379o-desmethyltramadolChemicalVariantAnnotationassociatedPK27082504
PA166157178rs12208357VariantVipGeneassociated
PA166157196rs34059508VariantVipGeneassociated
PA166157197rs34130495VariantVipGeneassociated14576340
PA166157216rs72552763VariantVipGeneassociated
PA443886Diabetes MellitusDiseaseClinicalAnnotationassociatedPD19381165, 19898263
PA443890Diabetes Mellitus, Type 2DiseaseClinicalAnnotationassociatedPKPD17111267, 22735389
PA443928DizzinessDiseaseVariantAnnotationassociatedPD23835420
PA443937Drug ToxicityDiseaseVariantAnnotationassociatedPD23835420
PA444065EpilepsyDiseaseClinicalAnnotationassociatedPKPD27610747
PA444354HeadacheDiseaseVariantAnnotationassociatedPD23835420
PA445048NauseaDiseaseVariantAnnotationassociatedPD23835420
PA445062NeoplasmsDiseaseClinicalAnnotationassociatedPKPD29427770, 30237583, 30713339
PA445208PainDiseaseVariantAnnotationassociatedPK27082504
PA445254Parkinson DiseaseDiseaseClinicalAnnotationassociatedPD
PA446171Leukemia, Myelogenous, Chronic, BCR-ABL PositiveDiseaseClinicalAnnotationassociatedPKPD24589908
PA448360amantadineChemicalClinicalAnnotationassociatedPD
PA449088codeineChemicalVariantAnnotationambiguousPKPD23835420
PA450163lamivudineChemicalPathwayassociated
PA450164lamotrigineChemicalClinicalAnnotationassociatedPKPD27610747
PA450213levodopaChemicalClinicalAnnotationassociatedPD
PA450395metforminChemicalClinicalAnnotation, Literature, MultilinkAnnotation, Pathway, VipGeneassociatedPKPD19536068, 19898263, 20690652, 21989078, 17111267, 17609683, 19381165, 19898263, 21989078, 22722338, 22735389, 24624919, 26700958, 27859023, 28380657, 28834135, 29352482
PA450550morphineChemicalVariantAnnotation, VipGeneassociatedPK23835420
PA451124proguanilChemicalVariantAnnotationassociatedPK29882324
PA451316selegilineChemicalClinicalAnnotationassociatedPD
PA451735tramadolChemicalClinicalAnnotation, VipGeneassociatedPK21562485
PA7000sorafenibChemicalMultilinkAnnotation, VipGeneassociated23532667

References

Pubmed IDYearTitleCitations
386053542024THOC7-AS1/OCT1/FSTL1 axis promotes EMT and serves as a therapeutic target in cutaneous squamous cell carcinoma.1
386053542024THOC7-AS1/OCT1/FSTL1 axis promotes EMT and serves as a therapeutic target in cutaneous squamous cell carcinoma.1
368538442023Pharmacogenetic impact of SLC22A1 gene variant rs628031 (G/A) in newly diagnosed Indian type 2 diabetes patients undergoing metformin monotherapy.0
378214932023Structural basis of promiscuous substrate transport by Organic Cation Transporter 1.4
368538442023Pharmacogenetic impact of SLC22A1 gene variant rs628031 (G/A) in newly diagnosed Indian type 2 diabetes patients undergoing metformin monotherapy.0
378214932023Structural basis of promiscuous substrate transport by Organic Cation Transporter 1.4
345450252022Association of SLC22A1 rs622342 and ATM rs11212617 polymorphisms with metformin efficacy in patients with type 2 diabetes.1
349023402022Molecular basis for stereoselective transport of fenoterol by the organic cation transporters 1 and 2.6
349272642022Genetic variants in SLC22A1 are related to serum lipid levels in Mexican women.1
352161202022Relationships between Inhibition, Transport and Enhanced Transport via the Organic Cation Transporter 1.7
354139902022OCT1-target neural gene PFN2 promotes tumor growth in androgen receptor-negative prostate cancer.6
354564162022The Role of SLC22A1 and Genomic Ancestry on Toxicity during Treatment in Children with Acute Lymphoblastic Leukemia of the Amazon Region.3
354699212022Amino acids in transmembrane helix 1 confer major functional differences between human and mouse orthologs of the polyspecific membrane transporter OCT1.5
345450252022Association of SLC22A1 rs622342 and ATM rs11212617 polymorphisms with metformin efficacy in patients with type 2 diabetes.1
349023402022Molecular basis for stereoselective transport of fenoterol by the organic cation transporters 1 and 2.6

Citation

Dessen P

SLC22A1 (solute carrier family 22 member 1)

Atlas Genet Cytogenet Oncol Haematol. 2010-05-01

Online version: http://atlasgeneticsoncology.org/gene/51461/slc22a1